論文 Publications

2016-

3. Othman, D. I. A.; Kitamura, M.* "Diazonaphthoquinones: Synthesis, Reactions and Applications", Heterocycles, DOI: 10.3987/REV-16-845.

2. Kitamura, M.*; Ishikawa, A.; Okauchi, T. "Synthesis, structure, and reaction of chiral 2-azidoimidazolinium salts: (7aS)-3-azido-5,6,7,7a-tetrahydro-2-[(1R)-1-phenylethyl]-1H-pyrrolo[1,2-c]imidazolium hexafluorophosphate and 2-azido-1,3-bis[(S)-1-phenylethyl]imidazolinium hexafluorophosphate" Tetrahedron Lett. 2016-

1. Kitamura, M.*; Fukuma, H.; Kobayashi, M.; Okayama, S.; Okauchi, T. "Axially Chiral Bifunctional 8,8??-Biquinolyl: Synthesis of 7,7??-Dihydroxymethyl-8,8??-biquinolyl via Pd-Catalyzed Double C-H Oxidation of 7,7??-Dimethyl-8,8??-biquinolyl" J. Org. Chem. 2016, 81, 3956-3960.

2011-2015

23. Kitamura, M.*; Takahashi, S.; Okauchi, T. "Rh-catalyzed Cyclization of 3-Aryloxycarbonyldiazonaphthoquinones for the Synthesis of beta-Phenylnaphthalene Lactones and Formal Synthesis of Pradimicinone" J. Org. Chem. 2015, 80, 8406-8416.

22 Kitamura, M.; Murakami, K. "Synthesis of 2-Azido-1,3-dimethylimidazolinium Hexafluorophosphate" Org. Synth. 2015, 92, 171-181.
21 Okauchi, T.*; Sata, N.; Urakawa, A.; Kitamura, M. "Unprecedented formation of hapto-4-(vinylketene)iron complexes from hapto-4-(diene)iron complexes and aromatic compounds in the presence of Lewis acid" Chem. Commun. 2015, 51, 8454-8456.

20 Kanetaka, H.; Koseki, Y.; Taira, J.; Umei, T.; Komatsu, H.; Sakamoto, H.; Gulten, G.; Sacchettini, J. C.; Kitamura, M.; Aoki, S.* "Discovery of InhA inhibitors with anti-mycobacterial activity through a matched molecular pair approach" Eur. J. Med. Chem. 2015, 94, 378-385.

19 Kitamura, M.*; Sakata, R.; Tashiro, N.; Ikegami, A.; Okauchi, T. "Synthesis of Diazonaphthoquinones from Naphthols by Diazo-transfer Reaction" Bull. Chem. Soc. Jpn. 2015, 88, 824-833.

18 Kitamura, M.; Yuasa, R.; Van Vranken, D. L.* "Synthesis of the Cyclic Prenylguanidine Nitensidine E using a Palladium-Catalyzed Carbenylative Amination" Tetrahedron Lett. 2015, 56, 3027-3031.

17 Kitamura, M.*; Kato, S.; Yano, M.; Tashiro, N.; Shiratake, Y.; Sando, M.; Okauchi, T. "Reagent for safe and efficient diazo-transfer to primary amines: 2-azido-1,3-dimethylimidazolinium hexafluorophosphate" Org. Biomol. Chem. 2014, 12, 4397-4406.

16 Kitamura, M.*; Kisanuki, M.; Kanemura, K.; Okauchi, T. "Pd(OAc)2-Catalyzed Macrocyclization of 1,2-Diazonaphthoquinones with Cyclic Ethers" Org. Lett. 2014, 16, 1554-1557.

15 Kitamura, M.*; Kubo, K.; Yoshinaga, S.; Matsuzaki, H.; Ezaki, K.; Matsuura, T.; Matsuura, D.; Fukuzumi, N.; Araki, K.; Narasaki, M. "Synthetic study of kosinostatin aglycone: Synthesis of BCDE rings using alkoxycarbonylmethylation of diazonaphthoquinone" Thetrahedron Lett. 2014, 55, 1653-1656.

14 北村 充 "安定なジアゾ移動剤の開発-グアニジノジアゾニウム塩の合成と反応" 有機合成化学協会誌, 2014, 72, 14-25.

13 Kitamura, M.*; Araki, K.; Matsuzaki, H.; Okauchi, T. "Rhodium-catalyzed Reaction of Diazonaphthoquinones and Enol Ethers: Synthesis of Dihydronaphthofuran Derivatives and alpha-Naphthyl Esters" Eur. J. Org. Chem. 2013, 5045-5049.

12 Kinjo, T.; Koseki, Y.; Kobayashi, M.; Yamada, A.; Morita, K.; Yamaguchi, K.; Tsurusawa, R.; Gulten, G.; Komatsu, H.; Sakamoto, H.; Sacchettini, J. C.; Kitamura, M.; Aoki, S.* "Identification of Compounds with Potential Antibacterial Activity against Mycobacterium through Structure-Based Drug Screening" J. Chem. Inf. Model. 2013, 53, 1200-1212.

11 Kitamura, M.*; Murakami, K.; Shiratake, Y.; Okauchi, T. "Synthesis of alpha-Arylcarboxylic Acid Amides from Enol Silyl Ether via Migratory-Amidation with 2-Azido-1,3-dimethylimidazolinium Hexafluorophosphate" Chem. Lett. 2013, 42, 691-693.

10 Kitamura, M.*; Tokuda, Y.; Tashiro, N.; Okauchi, T. "Cu(OAc)2-mediated Cross-coupling Reaction of Benzophenone N,N,N-Trimethylhydrazonium Salts and Aryl Boronic Acids" Aust. J. Chem. 2012, 65, 1687-1690.

9 Kitamura, M.*; Koga, T.; Yano, M.; Okauchi, T. "Direct Synthesis of Organic Azides from Alcohols using 2-Azido-1,3-dimethylimidazolinium Hexafluorophosphate" Synlett 2012, 1335-1338.

8 Kitamura, M.; Kisanuki, M.; Okauchi, T. "Synthesis of 1,2-Naphthalenediol Diacetates by Rhodium(II)-Catalyzed Reaction of 1,2-Diazonaphthoquinones with Acetic Anhydride" Eur. J. Org. Chem. 2012, 905-907.

7 Kitamura, M.*; Kisanuki, M.; Sakata, R.; Okauchi, T. "Pd(II)-Catalyzed Formal O-H Insertion Reactions of Diazonaphthoquinones to Acetic Acid: Synthesis of 1,2-Naphthalenediol Derivatives" Chem. Lett. 2011, 40, 1129-1131.

6 Kitamura, M.*; Sakata, R.; Matsumoto, T. "1-Diazonaphthalen-2(1H)-one" Acta Cryst. 2011, E67, o1951.

5 Kitamura, M.*; Miyagawa, S.; Okauchi, T. "Synthesis of alpha, alpha-diarylacetamides from benzyl aryl ketones using 2-azido-1,3-dimethylimidazolinium hexafluorophosphate" Tetrahedron Lett. 2011, 52, 3158-3161.

4 Kitamura, M.*; Sakata, R.; Okauchi, T. "Palladium-Catalyzed Cross-Coupling Reactions of 2-Diazonaphthoquinones with Arylboronic Acids" Tetrahedron Lett. 2011, 52, 1931-1933.

3 Kitamura, M.*; Tashiro, N.; Miyagawa, S. Okauchi, T. "2-Azido-1,3-dimethylimidazolinium Salts: Efficient Diazo-Transfer Reagents for 1,3-Dicarbonyl Compounds" Synthesis 2011, 1037-1044.

2 Kitamura, M.*; Moriyasu, Y.; Okauchi, T. "Synthesis of Isoindole Derivatives by Palladium-Catalyzed Domino Reaction of (2-Alkynyl)phenylketone O-Pentafluorobenzoyloximes" Synlett 2011, 643-646.

1 Kitamura, M.*; Yano, M.; Tashiro, N.; Miyagawa, S.; Sando, M.; Okauchi, T. "Direct Synthesis of Organic Azides from Primary Amines with 2-Azido-1,3-Dimethylimidazolinium Hexafluorophosphate" Eur. J. Org. Chem. 2011, 458-462.

2006-2010

15 Okauchi, T.; Kuramoto, K.; Kitamura, M. "Facile Preparation of Aryl Sulfides Using Palladium Catalysis under Mild Conditions" Synlett 2010, 2891-2894.

14 Kitamura, M.; Tashiro, N.; Sakata, R.; Okauchi, T. "Synthesis of Diazonaphthoquinones from Naphthols by Diazo-transfer Reaction
with 2-Azido-1,3-dimethylimidazolinium Chloride" Synlett 2010, 2503-2505.

13 Kitamura, M.; Shintaku, Y.; Kudo, D. "Low-valent zirconocene-mediated cyclization of gamma, delta-unsaturated oximes" Tetrahedron Lett. 2010, 51, 4890-4893.

12 Kitamura, M.; Kitahara, D.; Okauchi, T. "Enantioselective synthesis of alpha-benzylalanine using trans-3,4-dihydro-3,4-diaryldibenzo[c,g]phenanthrene-3,4-diols" Synlett 2010, 2097-2100.

11 Okauchi, T.; Teshima, T.; Kawakubo, H.; Kagimoto, K.; Sugahara, Y.; Kitamura, M. "CO Insertion in Lithiated Diene-Tricarbonyliron Complexes", Chem. Commun. 2010, 46, 5015-5017.

10 Kitamura, M.; Tashiro, N.; Takamoto, Y.; Okauchi, T. "Direct Synthesis of Acyl Azides from Carboxylic Acids Using 2-Azido-1,3-Dimethylimidazolinium Chloride" Chem. Lett. 2010, 39, 732-733.

9 Kitamura, M.; Shiomi, K.; Kitahara, D.; Yamamoto, Y. Okauchi, T. "Pinacol Coupling of 2,2'-Biaryldiketone: An Application for the Synthesis of Enantiopure 3,4-Dihydro-dibenzo-[c,g]-phenanthrene-3,4-diol Derivatives" Synlett 2010, 1359-1362.

8 Kitamura, M.; Tashiro, N; Okauchi, T. "Azido-1,3-dimethylimidazolinium Chloride: An Efficient Diazo Transfer Reagent for 1,3-Dicarbonyl Compounds" Synlett 2009, 2943-2944.

7 Kitamura, M.; Narasaka, K. "Catalytic Radicalcyclization of Oximes" Bull. Chem. Soc. Jpn. 200881, 539-547

6 Zaman, S.; Kitamura, M.; Abell, A. D. "Synthesis of 5-phenyl 2-functionalized pyrroles by amino Heck and tandem amino Heck carbonylation reactions" Aust. J. Chem. 2007, 60, 624-626.

5 Tamiya, M; Ohmori, K; Kitamura, M; Kato, H; Arai, T; Oorui, M ; Suzuki, K. "General synthesis route to benanomicin-pradimicin antibiotics" Chem. Eur. J. 2007, 13, 9791-9823.

4 Narasaka, K.; Kitamura, M. "Synthesis of azaheterocycles by one electron reduction of oximes" Arkivoc 2006, Part 7, 245-260.

3 Kitamura, M.; Ihara, Y.; Uera, K.; Narasaka, K. "Total Synthesis of Peduncularine", Bull. Chem. Soc. Jpn. 2006, 79, 1552-1560.

2 Chiba, S.; Kitamura, M.; Narasaka, K. "Synthesis of (-)-Sordarin" J. Am. Chem. Soc. 2006, 128,6931-6937.

1 Kitamura, M.; Kudo, D.; Narasaka, K. "Palladium(0)-catalyzed synthesis of pyridines from beta-acetoxy-gamma,delta-unsaturated ketone oximes" Arkivoc, 2006, iii, 148-162.

2000-2005

25 Ohmori, K.; Tamiya, M.; Kitamura, M.; Kato, H.; Oorui, M.; Suzuki, K. "Regio- and Stereocontrolled Total Synthesis of Benanomicin B", Angew. Chem., Int. Ed., 2005, 44, 3871-3874.

24 Tanaka, K.; Kitamura, M.; Narasaka, K., "Synthesis of a-Carbolines by Copper-Catalyzed Radical Cyclization of b-3-Indolyl Ketone O-Pentafluorobenzoyloximes", Bull. Chem. Soc. Jpn. 2005, 78,1659-1664.

23 Kitamura, M.; Mori, Y.; Narasaka, K. "Photochemical Radical Cyclization of g,d-Unsaturated Ketone Oximes to 3,4-Dihydro-2H-pyrroles" Tetrahedron Lett. 2005, 46, 2373-2376.

22 Zaman, S.; Kitamura, M.; Abell, A. D., "Synthesis of Trisubstituted Imidazoles by Palladium-Catalyzed Cyclization of O-Pentafluorobenzoylamidoximes: Application to Amino Acid Mimetics with a C-Terminal Imidazole"Org. Lett. 2005, 7, 609-611.

21 Kitamura, M.; Yanagisawa, H.; Yamane, M.; Narasaka, K. "Palladium(0)-Catalyzed Amino-Heck Reaction of gamma,delta-Uusaturated Ketone N,N,N-Trimethylhydrazonium Salts" Heterocycles 2005, 65, 273-277

20 Narasaka, K.; Kitamura, M. "Amination with Oximes" Eur. J. Org. Chem. 2005, 4505.

19 Kitamura, M.; Suga, T.; Chiba, S.; Narasaka, K. “Synthesis of Primary Amines by the Electrophilic Amination of Grignard Reagents with 1,3-Dioxolan-2-one O-Sulfonyloxime” Org. Lett. 2004, 6, 4619-4621.

18 Kitamura, M.; Chiba, S.; Narasaka, K.“Synthesis of (±)-Sordaricin” Chem. Lett. 2004, 33, 942-943.

17 Ando, K.; Kitamura, M.; Miura, K.; Narasaka, K., “Theoretical and Experimental Study on the In-Plane SN2 Type Substitution Reaction of Haloalkenes with Inversion of Configuration at Vinylic Carbon”Org. Lett. 2004, 6, 2461-2463.

16 Chiba, S.; Kitamura, M.; Saku, O.; Narasaka, K., “Synthesis of 1-Azaazulenes from Cycloheptatrienylmethyl Ketone O-Pentafluorobenzoyloximes by Palladium-Catalyzed Cyclization” Bull. Chem. Soc. Jpn. 2004, 77, 785-796.

15 Azemi, T.; Kitamura, M.; Narasaka, K., “Transformation of 1,5- and 1,6-Dienes by Hydrozirconation and Oxidation with Cerium(IV) Compounds“ Tetrahedron 2004, 60, 1339-1344.

14 Kitamura, M.; Yoshida, M.; Kikuchi, T.; Narasaka, K., “Synthesis of Quinolines and 2H-Dihydropyrroles by Nucleophilic Substitution at the Nitrogen Atom of Oxime Derivatives” Synthesis, 2003, 15, 2415-2426.

13 Yanagisawa, H.; Miura, K.; Kitamura, M.; Narasaka, K.; Ando K., “Intramolecular Substitution Reaction of Lithium Alkylidene Carbenoids: Regioselective Synthesis of Indenes” Bull. Chem. Soc. Jpn. 2003, 76, 2009-2026.

12 Yoshida, M; Kitamura, M.; Narasaka, K., “Synthesis of Dihydropyrrole and Pyrrole Derivatives by Radical Cyclization of g,d-Unsaturated Ketone O-Acetyloximes” Bull. Chem. Soc. Jpn. 2003, 76, 2003-2008.

11 Baldovini, N.; Kitamura, M.; Narasaka, K., "Amination of Arenes with N,N-Dimethyl-2-imidazolidinone O-Methoxyacetyloxime Nicolas”Chem. Lett. 2003, 548-549.

10 Zaman, S.; Kitamura, M.; Narasaka, K., "Synthesis of Polycyclic Imines by Palladium-Catalyzed Domino Cyclization of Di- and Trienyl Ketone O-Pentafluorobenzoyloximes" Bull. Chem. Soc. Jpn. 2003, 76, 1055-1062.

9 Kitamura, M.; Chiba, S; Narasaka, K., "Synthesis of Primary Amines and N-Methylamines by the Electrophilic Amination of Grignard Reagents with 2-Imidazolidinone O-Sulfonyloxime" Bull. Chem. Soc. Jpn. , 2003, 76, 1063-1070.

8 Kitamura, M.; Narasaka, K., "Synthesis of Aza-Heterocycles from Oximes by Amino-Heck Reaction" Chem. Rec. 2002, 2, 268-277.

7 Yanagisawa, H.; Miura, K.; Kitamura, M.; Narasaka, K.; Ando, K., "Intramolecular substitution reaction of alkylidene-lithium carbenoids: Regioselective synthesis of indenes" Helv. Chim. Acta 2002, 85, 3130-3135.

6 Ohmori, K.; Kitamura, M.; Ishikawa, Y.; Kato, H.; Oorui, M.; Suzuki, K., "Semi pinacol strategy for constructing B-ring of pradimicin-benanomicin antibiotics" Tetrahedron Lett. 2002, 43, 7023-7026.

5 Koganemaru, Y.; Kitamura, M.; Narasaka, K., "Synthesis of dihydropyrrole derivatives by copper-catalyzed cyclization of gamma,delta-unsaturated ketone O- methoxycarbonyloximes" Chem. Lett. 2002, 784-785.

4 Tsutsui, H.; Kitamura, M.; Narasaka, K., "Synthesis of pyrrole derivatives by palladium-catalyzed cyclization of gamma delta-unsaturated ketone O-pentafluorobenzoyloximes" Bull. Chem. Soc. Jpn. 2002, 75, 1451-1460.

3 Kitamura, M.; Chiba, S.; Saku, O.; Narasaka, K., "Palladium-catalyzed synthesis of 1-azaazulenes from cycloheptatrienylmethyl ketone O-pentafluorobenzoyl oximes" Chem. Lett. 2002, 606-607.

2 Yoshida, M.; Kitamura, M.; Narasaka, K., "Synthesis of 3,4-dihydro-2H-pyrroles from gamma,delta-unsaturated ketone O-acetyloximes" Chem. Lett. 2002, 144-145.

1 Kitamura, M.; Zaman, S.; Narasaka, K., "Synthesis of spiro imines from oximes by palladinm-catalyzed cascade reaction" Synlett 2001, 974-976.

1995-2000

5 Kitamura, M.; Ohmori, K.; Suzuki, K., “Divergent Behavior of Cobalt-Complexed Enyne Having a Leaving Group”Tetrahedron Lett. 1999, 40, 4563-4566.

4 Kitamura, M.; Ohmori, K.; Kawase, T.; Suzuki, K., “Total Synthesis of Pradimicinone, the Common Aglycon of the Pradimicin?Benanomicin Antibiotics”Angew. Chem. Int. Ed. 1999, 38, 1229-1232.

3 Ohmori, K.; Kitamura, M.; Suzuki, K., “From Axial Chirality to Central Chiralities: Pinacol Cyclization of 2,2'-Biaryldicarbaldehyde to trans-9,10-Dihydrophenanthrene-9,10-diol” Angew. Chem. Int. Ed. 1999, 38, 1226−1229.

2 Nagasawa, T.; Taya, K.; Kitamura, M.; Suzuki, K., “Novel Migrating Group in 1,2-Anionotropic Reactions: Cobalt Complexation Facilitates 1,2-Shift of Alkynyl Groups”J. Am. Chem. Soc. 1996, 118, 8949−8950.

1 Nagasawa, T.; Kitamura, M.; Suzuki, K., “Cobalt-Complexation Makes 2-(1-alkynyl)propenes Good Ene Donors in Carbonyl-Ene Reaction”Synlett 1995, 1183-1186.

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